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I-Eptifibastatide yonyango lwe-snary ye-Ackery Syndrome 188627-80-7

Inkcazo emfutshane:

Igama: Eptififatide

Inombolo ye-CAS: 188627-80-7

Ifomula yaseMolecila: C35H49O12O9S2

Ubunzima bemolekyuli: 831.96

Inombolo ye-einecs: 641-366-7-7

Ukuxinana: I-1.60 ± 0.1 g / cm3 (eqikelelweyo)

Iimeko zokugcina: Itywinwe ngowomileyo, gcina i-freezer, phantsi kwe-15 ° C


Iinkcukacha zemveliso

Iimpawu zeMveliso

Iinkcukacha zemveliso

Igama Eptifibatide
Inombolo ye-CAS Ngo-1886627-80-7
Ifomula yemolekyuli C35H491O9s2
Ubunzima bemolekyuli I-831.96
Inombolo ye-einecs I-641-366-7
Ukuxinana I-1.60 ± 0.1 g / cm3 (iqikelele)
Iimeko zokugcina Itywinwe kwi-freezer, engaphantsi kweminyaka eyi-100 ° C

Izithethantonye

I-EptifibaceSibibaceSibibaceribestalt; I-Eptifibatide, ePh-Gy-Asp-Tys-pro-pro-pro-pro-pro-pro-pro-pro-pro-pro-pro-pro-pro-pro-pro-pro-pro-pro-pro-pro-pro-pro-pro-pro-pro-pro-pro-pro-pro-pro-pro-pro-pro-pro-pro-pro-( nomethyl)-N2-(3-mercapto-1-oxopropyl-L-lysylglycyl-La-aspartyl-L-tryptophyl-L-prolyl-L-cysteinamide;MPA-HAR-GLY-ASP-TRP-PRO-CYS-NH2(DISULFIDEBRIDGE,MPA1-CYS6).

Iplatlet Gycoprotein Adagonist

I-Etifibatide (i-Medifililrilril) yi-InvespePide PillCepteide I-IIB / IIA I-Atchptor Antagorest, ethintela i-Argleregation kunye ne-thrombois kunye ne-thrombosis ngokuthintela indlela yokugqibela yendawo yokuhlala. Xa kuthelekiswa ne-monoclonn anticlonnika, i-Eptifibatide inamandla, engakumbi kunye nokubopha i-gpiib / iia ngenxa yobukho be-amino ye-amino of-acid eyodwa ye-Amino Acid. Ke ngoko, kufanele ukuba ibe nefuthe elilungileyo lonyango kunyango olungenelele kwi-syndrome ye-ofisi kangaka. I-Plalet Gycoprotein i-IIB / IIA I-IIA I-IIIA YABASEBENZI BABADALA ZENZIWE KAKHULU, KUNYE kwaye okwangoku kukho iintlobo ezi-3 zamalungiselelo anokusetyenziswa kwikliniki, i-Abciximab, eTirofiban. ). Akukho mava amancinci ekusebenziseni iplanti ye-Glycoprotein / IIA Recictor Achagonists eChina, kwaye amachiza akhoyo alinganiselwe kakhulu. Ichiza elinye kuphela, i-tirofiban hydrochloride, isemarikeni. Ke ngoko, i-gutelet entsha yePillcoprotein ye-Iib yaphuhliswa. / IIA IIIA I-AAGPONTS inyanzelekile. I-Eptififini yasekhaya yimveliso yokulinganisa eveliswe nguChengduonigio yebhayiloji yebhayoloji Cooogiolo

Ukwahlulahlula

Ukuhlelwa kweZiyobisi ze-antipalet

Iziyobisi ze-antipeletlet ze-antipalettilet zinokwenziwa malunga nezigaba ezintathu: 1. I-cycloossegegenasege-1 (i-COX-1) infiritors, njenge-aspirin. I-2. I-Ithintelo yePlanethi yePlanethi ebanjiwe yi-Adenosine Diphosphate (efana ne-clopidogrel, e-Prasugrel, njl. Njl.) Ukongeza, kukho I-Prostaglandin EP3 I-Infinitors, amaziko amatsha emichiza kunye neziqwengana zekhemikhali ezisandula ukukhululwa kumayeza e-China eTshayina.


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