Igama | Eptifibatide |
Inombolo ye-CAS | Ngo-1886627-80-7 |
Ifomula yemolekyuli | C35H491O9s2 |
Ubunzima bemolekyuli | I-831.96 |
Inombolo ye-einecs | I-641-366-7 |
Ukuxinana | I-1.60 ± 0.1 g / cm3 (iqikelele) |
Iimeko zokugcina | Itywinwe kwi-freezer, engaphantsi kweminyaka eyi-100 ° C |
I-EptifibaceSibibaceSibibaceribestalt; I-Eptifibatide, ePh-Gy-Asp-Tys-pro-pro-pro-pro-pro-pro-pro-pro-pro-pro-pro-pro-pro-pro-pro-pro-pro-pro-pro-pro-pro-pro-pro-pro-pro-pro-pro-pro-pro-pro-pro-pro-pro-pro-pro-pro-( nomethyl)-N2-(3-mercapto-1-oxopropyl-L-lysylglycyl-La-aspartyl-L-tryptophyl-L-prolyl-L-cysteinamide;MPA-HAR-GLY-ASP-TRP-PRO-CYS-NH2(DISULFIDEBRIDGE,MPA1-CYS6).
I-Etifibatide (i-Medifililrilril) yi-InvespePide PillCepteide I-IIB / IIA I-Atchptor Antagorest, ethintela i-Argleregation kunye ne-thrombois kunye ne-thrombosis ngokuthintela indlela yokugqibela yendawo yokuhlala. Xa kuthelekiswa ne-monoclonn anticlonnika, i-Eptifibatide inamandla, engakumbi kunye nokubopha i-gpiib / iia ngenxa yobukho be-amino ye-amino of-acid eyodwa ye-Amino Acid. Ke ngoko, kufanele ukuba ibe nefuthe elilungileyo lonyango kunyango olungenelele kwi-syndrome ye-ofisi kangaka. I-Plalet Gycoprotein i-IIB / IIA I-IIA I-IIIA YABASEBENZI BABADALA ZENZIWE KAKHULU, KUNYE kwaye okwangoku kukho iintlobo ezi-3 zamalungiselelo anokusetyenziswa kwikliniki, i-Abciximab, eTirofiban. ). Akukho mava amancinci ekusebenziseni iplanti ye-Glycoprotein / IIA Recictor Achagonists eChina, kwaye amachiza akhoyo alinganiselwe kakhulu. Ichiza elinye kuphela, i-tirofiban hydrochloride, isemarikeni. Ke ngoko, i-gutelet entsha yePillcoprotein ye-Iib yaphuhliswa. / IIA IIIA I-AAGPONTS inyanzelekile. I-Eptififini yasekhaya yimveliso yokulinganisa eveliswe nguChengduonigio yebhayiloji yebhayoloji Cooogiolo
Ukuhlelwa kweZiyobisi ze-antipalet
Iziyobisi ze-antipeletlet ze-antipalettilet zinokwenziwa malunga nezigaba ezintathu: 1. I-cycloossegegenasege-1 (i-COX-1) infiritors, njenge-aspirin. I-2. I-Ithintelo yePlanethi yePlanethi ebanjiwe yi-Adenosine Diphosphate (efana ne-clopidogrel, e-Prasugrel, njl. Njl.) Ukongeza, kukho I-Prostaglandin EP3 I-Infinitors, amaziko amatsha emichiza kunye neziqwengana zekhemikhali ezisandula ukukhululwa kumayeza e-China eTshayina.