Ilungu ngalinye elivela kwiqela lethu lengeniso yentsebenzo enkulu lixabisa iimfuno zabathengi kunye nonxibelelwano lwentlangano yeSampulu yaMahla ye-China Qgb Semi Automatic Aerosol Spray Can Filling Machine, Ukukhokela umkhwa wale ntsimi yinjongo yethu eqhubekayo. Ukubonelela ngempahla yodidi lokuqala yinjongo yethu. Ukwenza ixesha elide elihle, singathanda ukusebenzisana nabo bonke abahlobo basekhaya nakwamanye amazwe. Ukuba unomdla ngaphakathi kweemveliso zethu, akufanele ulinde ukudibana nathi.
Ilungu ngalinye elivela kwiqela lethu lengeniso yentsebenzo enkulu lixabisa iimfuno zabathengi kunye nonxibelelwano lwentlanganoUmatshini weAerosol, Umatshini wokutywina we-aerosol waseTshayina, Injongo yethu kukunceda abathengi baqonde iinjongo zabo. Besisenza iinzame ezinkulu zokufezekisa le meko yokuphumelela kwaye sikwamkela ngokunyanisekileyo ukuba usijoyine. Ngelizwi, xa usikhetha, ukhetha ubomi obugqibeleleyo. Wamkelekile ukutyelela umzi-mveliso wethu kwaye wamkele iodolo yakho! Ngemibuzo engaphezulu, akufanele ungathandabuzi ukuqhagamshelana nathi.
| CAS | 204656-20-2 | Ifomula yeemolekyuli | C172H265N43O51 |
| Ubunzima beMolekyuli | 3751.20 | Imbonakalo | Mhlophe |
| Imeko yoGcino | Ukumelana nokukhanya, i-2-8 degree | Iphakheji | I-aluminium foil bag / vial |
| Ubunyulu | ≥98% | Ezothutho | Cold Chain kunye nokuhanjiswa kogcino olupholileyo |
Uhlobo lwe-2 yeswekile
ILiraglutide iphucula ulawulo lweswekile yegazi. Iyanciphisa i-hyperglycemia enxulumene nokutya (kwiiyure ezingama-24 emva kokulawulwa) ngokunyusa i-insulin secretion (kuphela) xa ifunwa ngokunyusa amanqanaba eglucose, ukulibazisa ukukhutshwa kwesisu, kunye nokucinezela i-prandial glucagon secretion.
Ilungele izigulane ezineswekile yegazi engekalawuleki kakuhle emva kwedosi ephezulu enyanyezelweyo ye-metformin okanye i-sulfonylureas yodwa. Isetyenziswa ngokudibeneyo ne-metformin okanye i-sulfonylureas.
Isebenza ngendlela exhomekeke kwi-glucose, oku kuthetha ukuba iya kuvuselela i-insulin secretion kuphela xa amanqanaba eglucose yegazi ephezulu kunesiqhelo, ukukhusela "ukugqithiswa". Ngenxa yoko, kubonisa umngcipheko ongenakulinganiswa we-hypoglycemia.
Inamandla okuthintela i-apoptosis kunye nokuvuselela ukuvuselelwa kweeseli ze-beta (ezibonwa kwizifundo zezilwanyana).
Yehlisa umdla wokutya kwaye inqande ukufumana ubunzima bomzimba, njengoko kubonisiwe kuphononongo lwentloko ukuya entloko ngokuchasene ne-glimepiride.
Isenzo se-Pharmacological
I-Liraglutide yi-analog ye-GLP-1 ene-97% yokulandelelana kwe-homology kwi-GLP-1 yomntu, enokuthi ibophe kwaye ivule i-GLP-1 receptor. I-GLP-1 receptor ijolise kwi-GLP-1 yemveli, ihomoni ye-incretin engapheliyo ekhuthaza ukukhuselwa kwe-insulin exhomekeke kwi-insulin kwiiseli ze-pancreatic β. Ngokungafaniyo ne-GLP-1 yemveli, iiprofayili ze-pharmacokinetic kunye ne-pharmacodynamic ze-liraglutide ebantwini zilungele irejimeni yokudosa kube kanye yonke imihla. Emva kwesitofu se-subcutaneous, indlela yayo yesenzo sexesha elide ibandakanya: ukuzibandakanya ngokwakho okunciphisa ukufunxa; ukubophelela kwi-albumin; Uzinzo oluphezulu lwe-enzyme kwaye ngaloo ndlela ixesha elide lesiqingatha sobomi be-plasma.
Umsebenzi we-liraglutide ulungelelwaniswa yintsebenziswano ethile kunye ne-GLP-1 receptor, ekhokelela ekunyukeni kwe-cyclic adenosine monophosphate (cAMP). I-Liraglutide ivuselela ukukhuselwa kwe-insulin ngendlela exhomekeke kwi-glucose, ngelixa inciphisa ukukhutshwa kweglucagon ngokugqithisileyo ngendlela exhomekeke kwi-glucose.
Ngoko ke, xa i-glucose yegazi iphakama, i-insulin secretion ivuselelwe, ngelixa i-glucagon secretion ivinjelwe. Ngokwahlukileyo, i-liraglutide inciphisa ukukhuselwa kwe-insulin ngexesha le-hypoglycemia ngaphandle kokuchaphazela ukukhutshwa kweglucagon. Inkqubo ye-hypoglycemic ye-liraglutide ikwabandakanya ukongezwa kwexesha lokukhupha isisu. I-Liraglutide yehlisa ubunzima bomzimba kunye nobunzima bomzimba ngokunciphisa indlala kunye nokuthatha amandla.
Ilungu ngalinye elivela kwiqela lethu lengeniso yentsebenzo enkulu lixabisa iimfuno zabathengi kunye nonxibelelwano lwentlangano yeSampulu yaMahla ye-China Qgb Semi Automatic Aerosol Spray Can Filling Machine, Ukukhokela umkhwa wale ntsimi yinjongo yethu eqhubekayo. Ukubonelela ngempahla yodidi lokuqala yinjongo yethu. Ukwenza ixesha elide elihle, singathanda ukusebenzisana nabo bonke abahlobo basekhaya nakwamanye amazwe. Ukuba unomdla ngaphakathi kweemveliso zethu, akufanele ulinde ukudibana nathi.
Isampulu yasimahla yeUmatshini wokutywina we-aerosol waseTshayina, Umatshini weAerosol, Injongo yethu kukunceda abathengi baqonde iinjongo zabo. Besisenza iinzame ezinkulu zokufezekisa le meko yokuphumelela kwaye sikwamkela ngokunyanisekileyo ukuba usijoyine. Ngelizwi, xa usikhetha, ukhetha ubomi obugqibeleleyo. Wamkelekile ukutyelela umzi-mveliso wethu kwaye wamkele iodolo yakho! Ngemibuzo engaphezulu, akufanele ungathandabuzi ukuqhagamshelana nathi.