Igama | I-lekrorelin |
Inombolo ye-CAS | I-53714-5-0-0 |
Ifomula yemolekyuli | C59h84n16O12 |
Ubunzima bemolekyuli | I-1209.4 |
Inombolo ye-einecs | I-633-395-9-9 |
Ukujikeleza okuthile | D25 -31.7 ° (C = 1 kwi-1% ye-Acetic Acid) |
Ukuxinana | 1.44 ± 0.1 g / cm3 (eqikelelweyo) |
Imeko yokugcina | -15 ° C |
Ifom | Icocekile |
I-acididity ilunge | (pka) 9.82 ± 0.15 (iqikelelwe) |
Ukungathobeli kwamanzi | Inyibilikiswa emanzini nge-1mg / ml |
I-LH-RHLEUPLINE; I-levrolide; i-levrolide (yomntu); [i-leuprorelin; [D-Leu-Glymone-Nhetmoneum-nulymone-nul10, i-D-Leu6, pro -I-UNHETATD9) -UKREEINEINORONE-STE-Gly10, D-Leu6, i-DE-LOUICMPURORTEMORTONORTONORTONORTONO5, i-DE-LOU6
I-levrolide, Goserelin, i-Triprelin i-Nafarelin ngamachiza aliqela asetyenziswayo esetyenziswayo kwi-Ovari ukuba asuse umhlaza webele webele. . Oko kukuthi, i-gonadropin ikhuselwe kukuhla kwe-piruitary, okukhokelela ekunciphiseni okufanelekileyo kwi-hormone yesondo eyamkelwe yi-ovary.
I-levrollide yi-gonadropin-ukukhulula i-hormone (i-vrh) i-analog, ipeptide ye-Amino Acids. This product can effectively inhibit the function of the pituitary-gonadal system, the resistance to proteolytic enzymes and the affinity to the pituitary GnRH receptor are stronger than GnRH, and the activity of promoting the release of luteinizing hormone (LH) is about 20 times that of GnRH. Ikwanefuthe elinamandla lokuthintela i-pituitary-gonad isebenza kune-gnrh. Kwinqanaba lokuqala lonyango, i-follicle ivuselela i-holmone (fsh), i-LH, i-Androgen inyuke, emva koko, ngenxa yokupheliswa kwe-fetu, i-lh no-Estrogen okanye i-Androgen ithintelwe kwi-hormones yehomoni. Izifo zesondo (ezinje ngomhlaza ovuthuzayo, i-endometriosis, njl. Njl.) Yiba nefuthe lonyango.
Okwangoku, ityuwa ye-acetate ye-leparoide isetyenziswa ikakhulu ekliniki, kuba ukwenziwa kwe-leuptate ye-leuptate kuhlala kuzinzile kakhulu kubushushu begumbi. Ulwelo kufuneka lulahliwe. Ingasetyenziselwa ukuqiniswa kwencam yeziyobisi kwi-endometrios kunye ne-fibroine ye-fibroid, umhlaza wamabele ophambili we-humine, kunye nomhlaza webele, kunye ne-sporine yomhlaza, kunye nokungasebenzi kakuhle. Ingasetyenziselwa ukuchongwa ngaphambi kokufika kwe-femometrind, enokutyibilika ngokungqongqo, ukunciphisa i-Edema, kwaye inciphise ubunzima botyando.