I-Semaglutide ayiyona nje i-chiza yokulahlekelwa kwesisindo-lunyango oluyimpumelelo olujolise kwiingcambu ze-biological ezibangela ukukhuluphala.
1. Izenzo ebuchotsheni ukucinezela iSidlo
I-Semaglutide ilinganisa i-hormone yendalo ye-GLP-1, eyenza i-receptors isebenze kwi-hypothalamus-indawo yengqondo ejongene nokulawula indlala kunye nokuzala.
Iziphumo:
Yandisa ukuhlutha (ukuziva ugcwele)
Yehlisa indlala kunye nokunqwenela ukutya
Yehlisa ukutya okuqhutywa ngumvuzo (ukuthanda iswekile kunye nokutya okunekhalori ephezulu)
✅ Iziphumo: Ngokwendalo usebenzisa iikhalori ezimbalwa ngaphandle kokuziva uvinjwa.
2. Icothisa ukuKhupha kweGastric
I-Semaglutide inciphisa izinga apho ukutya kushiya isisu kwaye kungena emathunjini.
Iziphumo:
Yandisa imvakalelo yokuhlutha emva kokutya
Uzinzisa i-glucose spikes emva kokutya
Ithintela ukutya kakhulu kunye nokutya phakathi kokutya
✅ Isiphumo: Umzimba wakho uhlala wanelisekile ixesha elide, unciphisa ukuthathwa kwekhalori.
3. Ukuphucula ukuLawulwa kweSwekile yegazi
I-Semaglutide iphakamisa ukukhuselwa kwe-insulin xa iswekile yegazi iphezulu kwaye iyanciphisa ukukhululwa kwe-glucagon, ihomoni eyandisa iswekile yegazi.
Iziphumo:
Ukuphucula i-glucose metabolism
Yehlisa ukumelana ne-insulin (igalelo elikhulu ekugcineni amafutha)
Inqanda ukuphakama nokuhla kweswekile yegazi ebangela indlala
✅ Isiphumo: Indawo ezinzileyo yemetabolism exhasa ukutshiswa kwamafutha endaweni yokugcinwa kwamafutha.
4. Ikhuthaza uLahleko lweFat kwaye ikhusela i-Lean Muscle Mass
Ngokungafani neendlela zendabuko zokulahlekelwa kwesisindo ezinokubangela ukulahleka kwemisipha, i-Semaglutide inceda umzimba ukuba utshise amanqatha ngokukhethayo.
Iziphumo:
Yandisa i-fat oxidation (ukutshiswa kwamafutha)
Yehlisa i-visceral fat (ejikeleze izitho), edibene nesifo seswekile kunye nesifo senhliziyo
Igcina ubunzima bezihlunu ezibhityileyo ukuze umzimba ube sempilweni
✅ Isiphumo: Ukuncitshiswa kwexesha elide kwipesenti yamafutha omzimba kunye nokuphuculwa kwempilo yemetabolism.
Ubungqina beklinikhi
I-Semaglutide ibonise iziphumo ezingazange zibonwe ngaphambili kwizilingo zeklinikhi:
| Uvavanyo | Umthamo | Ubude bexesha | I-Avareji yokunciphisa umzimba |
|---|---|---|---|
| INYATHELO 1 | 2.4 mg ngeveki | Iiveki ezingama-68 | I-14.9% yobunzima bomzimba wonke |
| INYATHELO 4 | 2.4 mg ngeveki | Iiveki ezingama-48 | Ukulahleka kwesisindo okuqhubekayo emva kweeveki ze-20 zokusetyenziswa |
| INYATHELO 8 | 2.4 mg vs amanye amachiza e-GLP-1 | Intloko ukuya entloko | I-Semaglutide ivelise ukunciphisa okukhulu kwamafutha |
Ixesha lokuposa: Oct-23-2025
