Iimveliso
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CJC-1295
I-CJC-1295 API iveliswa kusetyenziswa iteknoloji yesigaba esiqinileyo se-peptide synthesis (SPPS) kwaye ihlanjululwe kusetyenziswa i-HPLC ukufezekisa ukucoceka okuphezulu kunye ne-batch-to-batch consistency.
Iimpawu zeMveliso:Ubunyulu ≥ 99%
Izinyibilikisi ezishiyekileyo ezisezantsi kunye neentsimbi ezinzima
Indlela ye-endotoxin-free, non-immunogenic synthesis
Ubungakanani obulungiselelweyo: mg ukuya kwikg
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NAD+
Iimpawu zeAPI:
Ukucoceka okuphezulu ≥99%
Pharmaceutical-grade NAD +
Imigangatho yokuvelisa efana ne-GMP
I-NAD + API ilungele ukusetyenziswa kwi-nutraceuticals, ii-injection, kunye nonyango oluphambili lwe-metabolic.
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I-Boc-Tyr(tBu)-Aib-Glu(OtBu)-Gly-OH
I-Boc-Tyr(tBu)-Aib-Glu(OtBu)-Gly-OHyitetrapeptide ekhuselweyo eqhele ukusetyenziswa kuphando lwe-peptide synthesis. Amaqela e-Boc (tert-butyloxycarbonyl) kunye ne-tBu (tert-butyl) asebenza njengamaqela akhuselayo ukuthintela ukusabela okusecaleni ngexesha lokudityaniswa kwekhonkco le-peptide. Ukufakwa kwe-Aib (α-aminoisobutyric acid) kunceda ukukhupha izakhiwo ze-helical kunye nokwandisa ukuzinza kwe-peptide. Olu landelelwano lwe-peptide lufundelwa amandla alo kuhlalutyo oluhambelanayo, ukusonga i-peptide, kwaye njengebhloko yokwakha ekuphuhliseni iipeptides ze-bioactive kunye nozinzo oluphuculweyo kunye neenkcukacha.
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Cagrilintide
I-Cagrilintide i-synthetic, i-amylin receptor agonist yexesha elide iphuhliswe ukunyangwa kokukhuluphala kunye nokuphazamiseka kwe-metabolic ezinxulumene nobunzima. Ngokulinganisa ihomoni yendalo i-amylin, inceda ukulawula ukutya, ukucotha kwesisu, kunye nokuphucula ukuhlutha. I-API yethu ephezulu ye-Cagrilintide API iveliswa ngokusebenzisa i-chemical synthesis kwaye idibana nemigangatho yemigangatho ye-pharmaceutical-grade, eyenza ifaneleke ukusetyenziswa kwiifom zokulawula ubunzima obuphezulu.
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Tesamorelin
I-Tesamorelin API isebenzisa itekhnoloji yenqanaba eliphezulu le-peptide synthesis (SPPS) kwaye inezi mpawu zilandelayo:
Ubunyulu ≥99% (HPLC)
Akukho i-endotoxin, iintsimbi ezinzima, izinyibilikisi ezishiyekileyo ezivavanyiweyo
Ukulandelelana kwe-amino acid kunye nesakhiwo esiqinisekiswe yi-LC-MS/NMR
Ukubonelela ngemveliso eyenziwe ngokwezifiso kwiigram ukuya kwiikhilogram -
Fmoc-Ile-Aib-OH
I-Fmoc-Ile-Aib-OH yibhloko yokwakha yeepeptide esetyenziswa kwi-soli-phase peptide synthesis (SPPS). Idibanisa i-isoleucine ekhuselweyo ye-Fmoc kunye ne-Aib (i-α-aminoisobutyric acid), i-amino acid engeyiyo yendalo eyenza i-helix iqine kunye nokuxhathisa i-protease.
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Fmoc-L-Lys[Eic(OtBu)-γ-Glu(OtBu)-AEEA-AEEA]-OH
I-Fmoc-L-Lys [Eic (OtBu)-γ-Glu (OtBu)-AEEA-AEEA] -OH yibhloko yokwakha i-amino acid esebenzayo eyenzelwe ukuhanjiswa kweziyobisi ezijoliswe kuyo kunye ne-bioconjugation. Ibonisa i-Eic (eicosanoid) i-moiety yokusebenzisana kwe-lipid, i-γ-Glu yokujolisa, kunye ne-AEEA spacers yokuguquguquka.
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Boc-Tyr(tBu)-Aib-OH
I-Boc-Tyr(tBu)-Aib-OH yibhloko yokwakha yeedipeptide ekhuselweyo esetyenziswa kwi-peptide synthesis, edibanisa i-Boc-protected tyrosine kunye ne-Aib (α-aminoisobutyric acid). Intsalela ye-Aib yongeza ukubunjwa kwe-helix kunye nokumelana ne-protease.
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Boc-His(Trt)-Ala-Glu(OtBu)-Gly-OH
I-Boc-His (Trt)-Ala-Glu (OtBu)-Gly-OH yiqhekeza le-tetrapeptide elikhuselweyo elisetyenziswe kwi-peptide synthesis yesigaba esiqinileyo (SPPS) kunye nophuhliso lweziyobisi ze-peptide. Ibandakanya amaqela akhuselayo kwi-orthogonal synthesis kunye neempawu zokulandelelana luncedo kwi-bioactive kunye ne-structural peptide design.
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I-Fmoc-Ls(Pal-Glu-OtBu)-OH
I-Fmoc-Lys(i-Pal-Glu-OtBu)-OH yibhloko ekhethekileyo ye-amino acid yokwakha eyenzelwe i-peptide-lipid conjugation. Ibonisa i-lysine ekhuselweyo ye-Fmoc kunye nekhonkco lecala le-palmitoyl-glutamate, ukuqinisa ubudlelwane be-membrane kunye ne-bioavailability.
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Fmoc-Yakhe-Aib-OH
I-Fmoc-His-Aib-OH yibhloko yokwakha yeepeptide esetyenziswa kwi-peptide synthesis, edibanisa i-Fmoc-protected histidine kunye ne-Aib (α-aminoisobutyric acid). I-Aib yazisa ukuqina kwe-conformational, iyenza ixabiseke ekuyileni i-helical kunye ne-stable peptides.
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Boc-His(Trt)-Aib-Glu(OtBu)-Gly-OH
I-Boc-His (Trt)-Aib-Glu (OtBu)-Gly-OH isiqwenga se-tetrapeptide ekhuselweyo esisetyenziswe kwi-peptide synthesis kunye nophuhliso lweziyobisi. Iqulethe amaqela asebenzayo akhuselweyo ngobuchule bokudibanisa i-stepwise kunye neempawu ze-Aib (α-aminoisobutyric acid) ukunyusa uzinzo lwe-helix kunye nobulukhuni be-conformational.
