Ukubambelela kwinkolelo "yokwenza izinto eziphezulu zoluhlu kunye nokwenza abahlobo kunye nabantu namhlanje abavela kwihlabathi lonke", sihlala sibeka umdla wabathengi kwindawo yokuqala yexabiso elicatshulweyo leChina Healthy Weight Loss CAS 96829-58-2 99% Bulk API Rimonbant CetilistatI-Orlistat, Ukusukela ekusekweni ngaphakathi kwiminyaka yoo-1990s, ngoku siye sakha inethiwekhi yethu yokuthengisa e-USA, eJamani, eAsia, nakumazwe amaninzi akuMbindi Mpuma. Sijonge ukufumana umboneleli okumgangatho ophezulu we-OEM yehlabathi jikelele kunye ne-aftermarket!
Ukubambelela kwinkolelo "yokwenza izinto eziphezulu kuluhlu kunye nokwenza abahlobo nabantu namhlanje abavela kwihlabathi liphela", sihlala sibeka umdla wabathengi kwindawo yokuqala.China 96829-58-2, I-Orlistat, Ngenkqubo yengxelo yokuthengisa ecokisekileyo yaseburhulumenteni kunye nomsebenzi onzima we-300 wabasebenzi abanezakhono, inkampani yethu iphuhlise zonke iintlobo zezisombululo ukusuka kudidi oluphezulu, udidi oluphakathi ukuya kudidi oluphantsi. Olu khetho lulonke lwezinto ezintle lunika abathengi bethu ukhetho olwahlukileyo. Ngaphandle koko, inkampani yethu inamathela kumgangatho ophezulu kunye nexabiso elifanelekileyo, kwaye sikunika iinkonzo ezilungileyo ze-OEM kwiimpawu ezininzi ezidumileyo.
| Igama | Leuprorelin |
| Inombolo yeCAS | 53714-56-0 |
| Ifomula yemolekyuli | I-C59H84N16O12 |
| Ubunzima bemolekyuli | 1209.4 |
| Inombolo ye-EINECS | 633-395-9 |
| Ukujikeleza okuthe ngqo | I-D25 -31.7 ° (c = 1 kwi-1% i-acetic acid) |
| Ukuxinana | 1.44±0.1 g/cm3(Kuxelwe kwangaphambili) |
| Imeko yokugcina | -15°C |
| Ifom | Icocekile |
| I-acidity coefficient | (pKa) 9.82±0.15 (Kuxelwe kwangaphambili) |
| Ukunyibilika kwamanzi | I-Soluble emanzini kwi-1mg / ml |
LH-RHLEUPROLIDE;LEUPROLIDE;LEUPROLIDE(HUMAN);LEUPRORELIN;[DES-GLY10,D-LEU6,PRO-NHET9]-LUTEINIZINGHORMONE-RELEASINGHORMONEHUMAN;(DES-GLY10,D-LEU6,PRO -NHET9)-LUTEINIZINGHORMONE-RELEASINGHORMONE;(DES-GLY10,D-LEU6,PRO-NHET9)-LUTEINIZINGHORMONE-REASINGFACTOR;[DES-GLY10,D-LEU6,PRO-NHET9]-LH-RH(UMNTU)
I-Leuprolide, i-goserelin, i-triprelin, kunye ne-nafarelin ngamachiza amaninzi aqhelekileyo asetyenziswa kwiklinikhi yokususa ii-ovari kunyango lomhlaza webele we-premenopausal kunye nomhlaza we-prostate. (ekubhekiswa kuyo njengeziyobisi ze-GnRH-a), amachiza e-GnRH-a ayafana ngesakhiwo kwi-GnRH kwaye akhuphisana ne-pituitary GnRH receptors. Oko kukuthi, i-gonadotropin ekhutshwe yi-pituitary iyancipha, ekhokelela ekunciphiseni okukhulu kwehomoni yesini efihliweyo yi-ovary.
I-Leuprolide yi-gonadotropin-releasing hormone (GnRH) analog, i-peptide eyenziwe nge-9 amino acids. Le mveliso inokuthintela ngokufanelekileyo umsebenzi wenkqubo ye-pituitary-gonadal, ukuchasana ne-proteolytic enzymes kunye nokuxhamla kwi-pituitary GnRH receptor yomelele kune-GnRH, kwaye umsebenzi wokukhuthaza ukukhululwa kwe-hormone ye-luteinizing (LH) malunga namaxesha angama-20 kwi-GnRH. Ikwanayo nefuthe elinamandla lokuthintela ukusebenza kwe-pituitary-gonad kune-GnRH. Kwinqanaba lokuqala lokonyango, i-follicle stimulating hormone (FSH), i-LH, i-estrogen okanye i-androgen inokunyuswa okwethutyana, kwaye ke, ngenxa yokuncipha kokuphendula kwe-pituitary gland, ukukhutshwa kwe-FSH, i-LH kunye ne-estrogen okanye i-androgen ivinjelwe, okubangelwa ukuxhomekeka kwi-hormone yesini. Izifo zesondo (ezifana nomhlaza wesifo seprotate, i-endometriosis, njl.) zinefuthe lonyango.
Okwangoku, ityuwa ye-acetate ye-leuprolide isetyenziswa kakhulu kwikliniki, kuba ukusebenza kwe-acetate ye-leuprolide kuzinzile kwiqondo lokushisa. Ulwelo kufuneka ilahlwe. Ingasetyenziselwa unyango lokuthenwa kweyeza le-endometriosis kunye ne-uterine fibroids, ukufikisa okusembindini, umhlaza wamabele we-premenopausal kunye nomhlaza wesibeleko, kunye nokopha kwe-uterine esebenzayo echaseneyo okanye engasebenziyo kunyango lwe-hormone eqhelekileyo. Isenokusetyenziswa njenge-premedication phambi kwe-endometrial resection, enokuthi icuthe ngokulinganayo i-endometrium, inciphise i-edema, kwaye inciphise ubunzima botyando. Ukunamathela kwinkolelo "yokwenza izinto eziphezulu zoluhlu kunye nokwenza abahlobo kunye nabantu namhlanje abavela kwihlabathi liphela", siqhele ukubeka umdla wabathengi kwindawo yokuqala ngexabiso elicatshulweyo le-China Healthy Weight 92 CAS 98 Los 98 Los98 I-API Rimonbant Cetilistat Orlistat, Ukususela ekusekweni ngaphakathi kwi-1990s yokuqala, ngoku siye sakha inethiwekhi yethu yokuthengisa e-USA, eJamani, e-Asia, nakwamanye amazwe amaninzi akuMbindi Mpuma. Sijonge ukufumana umboneleli okumgangatho ophezulu we-OEM yehlabathi jikelele kunye ne-aftermarket!
Ixabiso elicatshulweyo leChina 96829-58-2, I-Orlistat, Ngenkqubo ye-state-of-art yokuthengisa ngokucokisekileyo kunye nomsebenzi onzima we-300 wabasebenzi abanezakhono, inkampani yethu iphuhlise zonke iintlobo zezisombululo ezivela kwiklasi ephezulu, iklasi ephakathi ukuya kwiklasi ephantsi. Olu khetho lulonke lwezinto ezintle lunika abathengi bethu ukhetho olwahlukileyo. Ngaphandle koko, inkampani yethu inamathela kumgangatho ophezulu kunye nexabiso elifanelekileyo, kwaye sikunika iinkonzo ezilungileyo ze-OEM kwiimpawu ezininzi ezidumileyo.