Glucagon API
IGlucagon yihomoni yendalo ye-peptide esetyenziswa njengonyango olungxamisekileyo kwi-hypoglycemia enzima kwaye ifundelwe indima yayo kulawulo lwe-metabolic, ukuncipha kobunzima, kunye noxilongo lokwetyisa.
Inkqubo kunye noPhando:
IGlucagon ibophelela kwi-glucagon receptor (GCGR) esibindini, ivuselela:
Ukuqhekeka kweGlycogen ukunyusa iswekile yegazi
I-Lipolysis kunye nokuhlanganiswa kwamandla
Ukumodareyitha kwe-gastrointestinal motility (isetyenziswa kwi-radiology)
Kwakhona kujongwa ngokukhuluphala, uhlobo lwe-2 yeswekile, kunye ne-agonists ezimbini / ezintathu zonyango kunye ne-GLP-1 kunye ne-GIP.
Iimpawu ze-API (iQela leGentolex):
Ipeptide yococeko oluphezulu (≥99%)
Iveliswe nge-soli-phase peptide synthesis (SPPS)
Umgangatho ofana ne-GMP
Ifanelekile kwizitofu kunye neekhithi zongxamiseko
IGlucagon API ibalulekile kuhlangulo lwe-hypoglycemia, ukucinga ngoxilongo, kunye nophando lwe-metabolic disorder.