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Teriparatide Acetate API for Osteoporosis CAS NO.52232-67-4

Inkcazelo emfutshane:

I-Teriparatide yi-synthetic 34-peptide, i-1-34 amino acid fragment ye-hormone ye-parathyroid ye-PTH, eyi-biologically esebenzayo ye-N-terminal yengingqi ye-84 amino acids endogenous parathyroid hormone PTH.Iimpawu ze-immunological kunye ne-biological zale mveliso zifana ncakasana ne-endogenous parathyroid hormone PTH kunye ne-bovine parathyroid hormone PTH (bPTH).


Iinkcukacha zeMveliso

Iithegi zeMveliso

Iinkcukacha zeMveliso

Igama I-Teriparatide Acetate
Inombolo yeCas. 52232-67-4Imolekyuli
Ifomula C181h291n55o51s2
Imbonakalo mhlophe ukuya kumhlophe
Ixesha lokuzisa Ulungile kwi-Stock
Iphakheji Isikhwama seAluminiyam yeFoil
Ubunyulu ≥98%
Ugcino I-2-8 degree
Ezothutho Ikhonkco elibandayo kunye nokuhanjiswa okupholileyo kokugcinwa

Izithethantonye

I-PARATHYROIDHORMONEHUMAN: I-FRAGMENT1-34;I-PARATHYROIDHORMONE(UMNTU,1-34);I-PARATHYROIDHORMONE (1-34), UMNTU;PTH (1-34) (UMNTU);I-PTH(UMNTU,1-34);I-TERIPARATIDE;I-Teriparatide acetate.

Umsebenzi

I-Teriparatide inokulamla i-metabolism yamathambo ngokuthintela i-osteoblast apoptosis, isebenze iiseli zamathambo, kunye nokuphucula ukwahlula kwe-osteoblast.Ngaphakathi ivuselela i-PHT-I receptor kumphezulu we-osteoblasts, iiseli zethambo kunye neeseli ze-stromal stem ze-bone umongo ngokulawula i-adenylate cyclase-cyclic adenosine monophosphate-protein kinase Indlela yokukhuthaza ukuhlukana kwe-osteoblast kunye nokwandisa ubomi beseli ye-osteogenesis;Ukuvuselela ukwanda kwemigca yeeseli ze-osteoblast ngokusebenzisa i-phosphate C-cytoplasmic calcium-protein Chemicalbook kinase C indlela yokubonisa;Ngokuthintela umsebenzi wokuguqulwa kwe-PPARγ, kunciphisa ukuhlukana kweeseli ze-stromal kumgca we-adipocyte kunye nokwandisa inani le-osteoblasts;Ukulawula ngokungathanga ngqo ukukhula kwamathambo ngokulawula i-cytokines, umzekelo, i-iGF-1 inokunyanzelwa ukuba ibophe i-osteoblasts, ngaloo ndlela ikhuthaza ukubunjwa kwamathambo;

Inkqubo yokubunjwa kwamathambo ilawulwa yindlela yokubonisa iWnt, ngaloo ndlela yandisa ukubunjwa kwamathambo.

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