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I-Micafungin ye-antifungal kunye ne-antiviral

Inkcazelo emfutshane:

Igama: Micafungin

Inombolo ye-CAS: 235114-32-6

Ifomula yemolekyuli: C56H71N9O23S

Ubunzima bemolekyuli: 1270.28

Inombolo ye-EINECS: 1806241-263-5


Iinkcukacha zeMveliso

Iithegi zeMveliso

Iinkcukacha zeMveliso

Igama Micafungin
inombolo yeCAS 235114-32-6
Ifomula yemolekyuli I-C56H71N9O23S
Ubunzima bemolekyuli 1270.28
Inombolo ye-EINECS 1806241-263-5

I-Clinical Pharmacology

Le mveliso yeyokufakwa kwi-intravenous.I-concentration ye-plasma ifikelela kwinqanaba eliphezulu ekupheleni kokunyuswa, kwaye ukuphelisa i-half-life yi-13.9 iiyure.Ukuxinwa kwe-micafungin kwimiphunga, isibindi, i-spleen kunye nezicubu zezintso yeyona iphakamileyo, kodwa ayifumanekanga kwi-cerebrospinal fluid.Emva kokufakwa kwi-intravenous, i-metabolized ikakhulu esibindini kwaye ikhutshwe kwindle kunye nomchamo.

Umsebenzi

I-dose ephakanyisiweyo yonyango lwe-candidiasis ye-esophageal yi-150 mg ngosuku, kwaye i-dose ephakanyisiweyo yokuthintela usulelo lwe-Candida kwizigulane ze-hematopoietic stem cell transplant yi-50 mg ngosuku.Ngokutsho kwedatha yeklinikhi ekhoyo, umyinge wonyango okanye uthintelo lwezifo ezibini ezingentla ziyi-15 iintsuku kunye neentsuku ze-19, ngokulandelanayo.Iyeza lilungiswe kwaye lihlanjululwe nge-saline eqhelekileyo okanye i-5% ye-dextrose injection.Ixesha lokulawula kufuneka libe ubuncinane iyure eli-1, ngaphandle koko kulula ukuvelisa ukusabela okubi.

Ukunxibelelana kwezamayeza

Incopho yoxinaniso lwe-plasma ye-nifedipine inokunyuswa ngama-42%, kwaye ukuba kuyimfuneko, cinga ukunciphisa umthamo we-nifedipine okanye ukuyeka ichiza.Ummandla ophantsi kwe-plasma yoxinaniso lwegophe ye-anti-organ rejection drug Sirolimus inyuke nge-21%, kwaye ukuncipha kwethamo le-sirolimus kufuneka kuthathelwe ingqalelo njengento efanelekileyo.Amachiza e-Antifungal, i-pharmacology yeklinikhi, ukusetyenziswa, ukusabela okubi, njl njl. ye-micafungin

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